SCHEMBL28010992

SCHEMBL28010992

OC1=CCCc2ncccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.47
TBXAS1 P24557 3/20 0.47
KDM4E B2RXH2 2/20 0.33
TDP1 Q9NUW8 2/20 0.32
KMT2A Q03164 2/20 0.32
TDP2 O95551 1/20 0.32
NSD2 O96028 1/20 0.32
ABL1 P00519 1/20 0.32
PLCG1 P19174 1/20 0.32
CES1 P23141 1/20 0.32
PAX8 Q06710 1/20 0.32
RIN1 Q13671 1/20 0.32
MEN1 O00255 1/20 0.32
THRB P10828 1/20 0.32
BLM P54132 1/20 0.32
GAA P10253 1/20 0.32
MAPK14 Q16539 2/20 0.32
MMP2 P08253 2/20 0.31
TSHR P16473 2/20 0.31
GMNN O75496 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27549267 0.98 CYP19A1 (0.46) CYP19A1TBXAS1KDM4ETDP1KMT2A
SCHEMBL12459199 0.77 CYP19A1 (0.47) CYP19A1TBXAS1KDM4ETDP1KMT2A
SCHEMBL27890627 0.77 CYP19A1 (0.47) CYP19A1TBXAS1KDM4ETDP1KMT2A
SCHEMBL22579802 0.74 TDP1 (0.42) CYP19A1TBXAS1KDM4ETDP1KMT2A
SCHEMBL24097109 0.73 CYP19A1 (0.43) CYP19A1TBXAS1PDK2CYP1A2
SCHEMBL3860294 0.73 CYP19A1 (0.43) CYP19A1TBXAS1CYP3A4HTTALDH1A1
SCHEMBL28228601 0.71 PDE5A (0.40) CYP19A1TBXAS1KDM4ETDP1TSHR
SCHEMBL28125072 0.71 L3MBTL1 (0.40) CYP19A1TBXAS1KDM4ETDP1TDP2
SCHEMBL3861319 0.69 CYP3A4 (0.48) CYP19A1TBXAS1MAPK14CYP3A4CYP1A2
SCHEMBL16550205 0.69 HRH1 (0.36) KDM4ETDP1KMT2ATDP2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103221405-B Substituted pyridine compound DAIICHI SANKYO CO LTD 2015-04-22 CN claimed
CN-103221405-B Substituted pyridine compound DAIICHI SANKYO CO LTD 2015-04-22 CN disclosed