Methylamine

Methylamine

SCHEMBL28014455

CN.CN.CN.O=C1Cc2ccc(F)cc2N1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AHR P35869 4/20 0.56
CMA1 P23946 2/20 0.56
EIF2AK2 P19525 1/20 0.54
PDK2 Q15119 1/20 0.48
TDP2 O95551 1/20 0.48
HTR5A P47898 2/20 0.47
CRBN Q96SW2 3/20 0.47
HDAC3 O15379 1/20 0.45
MAOB P27338 2/20 0.44
GRIA1 P42261 1/20 0.43
CACNG8 Q8WXS5 1/20 0.43
PGR P06401 1/20 0.42
CA9 Q16790 1/20 0.42
SMYD3 Q9H7B4 1/20 0.42
KDM1A O60341 1/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30648196 0.94 AHR (0.61) AHRCMA1EIF2AK2PDK2TDP2
SCHEMBL260027 0.94 AHR (0.61) AHRCMA1EIF2AK2PDK2TDP2
SCHEMBL7717893 0.93 AHR (0.59) AHRCMA1EIF2AK2PDK2TDP2
SCHEMBL5843103 0.82 CRBN (0.57) AHRCMA1EIF2AK2PDK2TDP2
Methylamine SCHEMBL28015139 0.80 CA9 (0.66) AHRCMA1EIF2AK2PDK2TDP2
SCHEMBL152963 0.79 AHR (0.61) AHRCMA1PDK2TDP2HTR5A
Methylamine SCHEMBL27858404 0.79 AHR (0.89) AHRCMA1EIF2AK2PDK2TDP2
SCHEMBL29754281 0.78 CA9 (0.62) HTR5ACRBNMAOBCA9
SCHEMBL4102521 0.78 CA9 (0.62) HTR5ACRBNMAOBCA9
SCHEMBL7505614 0.76 MAPT (0.59) AHRCMA1HTR5ACRBNCA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104619701-A 2-oxo-2,3-dihydro-indoles for the treatment of cns disorders HOFFMANN LA ROCHE 2015-05-13 CN disclosed