SCHEMBL28014875

SCHEMBL28014875

CC(C)(C)NC(=O)OC1CCN(C(=O)CC#N)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.43
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
JAK2 O60674 11/20 0.36
JAK3 P52333 11/20 0.36
ROCK1 Q13464 3/20 0.36
PKN2 Q16513 3/20 0.36
LRRK2 Q5S007 3/20 0.36
LCK P06239 2/20 0.36
RET P07949 2/20 0.36
KDR P35968 2/20 0.36
CAMK1D Q8IU85 2/20 0.36
PRKACA P17612 1/20 0.36
LTK P29376 1/20 0.36
GSK3A P49840 1/20 0.36
PRKX P51817 1/20 0.36
PIK3CD O00329 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28025455 0.84 DPP4 (0.39) DPP4PIK3CDSMN1; SMN2LMNA
SCHEMBL27955404 0.79 SMN1; SMN2 (0.39) DPP4ALDH1A1MAPTPIK3CDSMN1; SMN2
SCHEMBL23895694 0.78 JAK3 (0.41) MEN1ALDH1A1MAPTKMT2AJAK2
SCHEMBL17308196 0.78 JAK3 (0.41) MEN1ALDH1A1MAPTKMT2AJAK2
SCHEMBL30497351 0.78 JAK3 (0.41) MEN1ALDH1A1MAPTKMT2AJAK2
SCHEMBL22388263 0.75 JAK3 (0.39) MEN1ALDH1A1MAPTKMT2AJAK2
SCHEMBL27756928 0.75 ALDH1A1 (0.51) DPP4MEN1ALDH1A1MAPTKMT2A
SCHEMBL29143876 0.75 EPHX2 (0.43) DPP4MEN1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL17320497 0.75 PIK3CD (0.41) DPP4MEN1ALDH1A1MAPTKMT2A
SCHEMBL17306173 0.74 IRAK4 (0.39) MEN1ALDH1A1MAPTKMT2AJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104650092-B Substituted heteroaryl compound and combinations thereof and purposes 广东东阳光药业有限公司 2017-11-10 CN disclosed
CN-104650092-A Substituted ceteroary compound as well as composition and application thereof GUANGDONG HEC PHARMACEUTICAL 2015-05-27 CN disclosed