SCHEMBL28015207

SCHEMBL28015207

C=C(C(=O)OC)c1c(N)cccc1F

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.44
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
CRBN Q96SW2 1/20 0.41
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CFTR P13569 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HDAC1 Q13547 1/20 0.38
PREP P48147 1/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28094324 0.88 POLB (0.50) POLBCES2CES1RAB9AKMT2A
SCHEMBL27757319 0.82 CA12 (0.52) POLBCES2CES1RAB9AKMT2A
SCHEMBL1489210 0.80 CA12 (0.52) POLBCES2CES1CRBNRAB9A
SCHEMBL28259615 0.77 POLB (0.42) POLBCES2CES1RAB9AALDH1A1
SCHEMBL6989228 0.74 CES2 (0.46) POLBCES2CES1CRBNRAB9A
SCHEMBL28350547 0.74 NPC1 (0.43) POLBRAB9AALDH1A1KMT2AMEN1
SCHEMBL10441887 0.73 CES2 (0.64) POLBCES2CES1RAB9AKMT2A
SCHEMBL14454258 0.73 CES2 (0.52) POLBCES2CES1CRBNHDAC1
SCHEMBL4089662 0.73 CES2 (0.52) CES2CES1CRBNALDH1A1HDAC1
SCHEMBL6989232 0.73 CES2 (0.40) POLBCES2CES1CRBNRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104619694-A Azetidine and piperidine compounds useful as PDE10 inhibitors AMGEN INC 2015-05-13 CN disclosed