SCHEMBL28016276

SCHEMBL28016276

NCc1ccc(C(=O)n2nc(-c3ccccc3)cc2NCc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 9/20 0.56
HTT P42858 2/20 0.45
RAB9A P51151 2/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
CYP2C9 P11712 1/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
KLKB1 P03952 4/20 0.44
KLK1 P06870 2/20 0.44
CFD P00746 1/20 0.44
PHGDH O43175 1/20 0.43
MAPT P10636 4/20 0.43
KDM4E B2RXH2 2/20 0.43
VCP P55072 1/20 0.43
THRB P10828 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28016807 0.92 F2 (0.53) F2HTTRAB9AMEN1ALDH1A1
SCHEMBL28016154 0.92 F2 (0.57) F2ALDH1A1LMNAPOLBKMT2A
SCHEMBL2569658 0.91 F2 (0.60) F2HTTRAB9AMEN1ALDH1A1
SCHEMBL2566670 0.87 F2 (0.69) F2RAB9APOLBKMT2AKLKB1
SCHEMBL2568116 0.87 F2 (0.57) F2HTTRAB9AMEN1ALDH1A1
SCHEMBL2561986 0.87 KLKB1 (0.55) F2HTTRAB9AMEN1ALDH1A1
SCHEMBL2569334 0.86 KLKB1 (0.57) F2KLKB1KLK1MAPTTHRB
SCHEMBL2563383 0.85 F2 (0.72) F2RAB9AALDH1A1LMNAPOLB
SCHEMBL2555846 0.85 F2 (0.57) F2RAB9AMEN1CYP1A2POLB
SCHEMBL2568165 0.85 F2 (0.60) F2HTTMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102918034-B Polysubstituted aromatic compounds as inhibitors of thrombin VERSEON CORP 2015-06-03 CN claimed