SCHEMBL28016807

SCHEMBL28016807

NCc1cccc(C(=O)n2nc(-c3ccccc3)cc2NCc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 8/20 0.53
CFD P00746 1/20 0.48
HTT P42858 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 2/20 0.45
THRB P10828 2/20 0.45
KLKB1 P03952 3/20 0.43
KLK1 P06870 1/20 0.43
LDHA P00338 1/20 0.42
LDHB P07195 1/20 0.42
TP53 P04637 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.40
GRM5 P41594 1/20 0.40
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28016276 0.92 F2 (0.56) F2CFDHTTKDM4EMAPT
SCHEMBL28016243 0.92 MAPT (0.56) F2KDM4EMAPTTHRBKLKB1
SCHEMBL2569658 0.90 F2 (0.60) F2HTTKDM4EMAPTTHRB
SCHEMBL14687509 0.87 MAPT (0.59) F2HTTKDM4EMAPTTHRB
SCHEMBL14688360 0.87 MAPT (0.59) F2HTTKDM4EMAPTTHRB
SCHEMBL14688774 0.87 F2 (0.61) F2HTTKDM4EMAPTTHRB
SCHEMBL28016154 0.84 F2 (0.57) F2KDM4EMAPTTHRBKLKB1
SCHEMBL2564978 0.84 F2 (0.53) F2HTTKDM4EMAPTTHRB
SCHEMBL14688467 0.84 POLB (0.55) F2MAPTKLKB1KLK1TP53
SCHEMBL2573709 0.84 GRM5 (0.55) F2HTTKDM4EMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102918034-B Polysubstituted aromatic compounds as inhibitors of thrombin VERSEON CORP 2015-06-03 CN claimed