SCHEMBL28017154

SCHEMBL28017154

COc1cccc(/C=C/C(=O)c2ccc3nc(C)[nH]c(=O)c3c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.58
BCHE P06276 1/20 0.58
LMNA P02545 3/20 0.57
KDM4E B2RXH2 1/20 0.57
HSD17B10 Q99714 1/20 0.57
ALDH1A1 P00352 2/20 0.55
CYP1A1 P04798 4/20 0.55
CYP1A2 P05177 4/20 0.55
CYP1B1 Q16678 4/20 0.55
CYP2D6 P10635 3/20 0.55
IP6K1 Q92551 1/20 0.54
MAPT P10636 2/20 0.53
CYP3A4 P08684 3/20 0.52
ABCG2 Q9UNQ0 4/20 0.52
ABCB1 P08183 2/20 0.52
P4HB P07237 1/20 0.49
TUBB4A P04350 1/20 0.49
TUBB P07437 1/20 0.49
TUBA3C P0DPH7 1/20 0.49
TUBA1B P68363 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819521 0.87 IP6K1 (0.67) MAOBBCHELMNAKDM4EHSD17B10
SCHEMBL28819517 0.87 IP6K1 (0.67) MAOBBCHELMNAKDM4EHSD17B10
SCHEMBL28017664 0.81 MAPT (0.57) MAOBBCHELMNAKDM4EHSD17B10
SCHEMBL28017674 0.80 IP6K1 (0.56) MAOBHSD17B10CYP1B1IP6K1ABCG2
SCHEMBL28819820 0.80 IP6K1 (0.56) MAOBLMNAKDM4EHSD17B10ALDH1A1
SCHEMBL28017127 0.80 IP6K1 (0.56) MAOBLMNAKDM4EHSD17B10ALDH1A1
SCHEMBL28017665 0.78 IP6K1 (0.54) MAOBLMNAHSD17B10ALDH1A1CYP1B1
SCHEMBL28017668 0.78 IP6K1 (0.54) MAOBLMNAHSD17B10ALDH1A1CYP1B1
SCHEMBL28017157 0.77 IP6K1 (0.53) MAOBLMNAKDM4EHSD17B10ALDH1A1
SCHEMBL31298986 0.76 MAOB (0.86) MAOBBCHELMNAALDH1A1CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104803927-A Chalcone analogue containing 2-methyl-4-oxo-quinazoline-6-base, and preparation method and application thereof UNIV CAPITAL NORMAL 2015-07-29 CN disclosed