SCHEMBL28017608

SCHEMBL28017608

CC(F)(F)c1cnc[nH]c1=O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.38
ALDH1A1 P00352 3/20 0.37
FKBP5 Q13451 1/20 0.37
HPGD P15428 1/20 0.35
SCN9A Q15858 1/20 0.33
HRH3 Q9Y5N1 5/20 0.32
HRH4 Q9H3N8 4/20 0.32
PDPK1 O15530 1/20 0.31
KDM4A O75164 1/20 0.31
KDM4B O94953 1/20 0.31
KDM5C P41229 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
KDM3A Q9Y4C1 1/20 0.31
CYP17A1 P05093 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28018128 0.83 PARP1 (0.43) PARP1ALDH1A1FKBP5SCN9AHRH3
SCHEMBL24880089 0.80 ALDH1A1 (0.37) ALDH1A1FKBP5HPGDCYP17A1CYP3A4
SCHEMBL26064901 0.70 HRH3 (0.40) HRH3HRH4CYP3A4
SCHEMBL849426 0.67
SCHEMBL312270 0.67
SCHEMBL25435625 0.67 ALDH1A1 (0.39) ALDH1A1FKBP5HPGDHRH3KDM4A
Fluoxidine SCHEMBL1369498 0.67
Bromide SCHEMBL1938531 0.66
SCHEMBL22139827 0.63 HPGD (0.50) PARP1ALDH1A1HPGDPDPK1KDM5B
SCHEMBL1771094 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104822670-A 5-phenoxy-3h-pyrimidin-4-one derivatives and their use as HIV reverse transcriptase inhibitors MERCK SHARP & DOHME 2015-08-05 CN disclosed