SCHEMBL28019207

SCHEMBL28019207

CS(=O)(=O)c1ccccc1C(O)C=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
BCAT2 O15382 1/20 0.37
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
KCNH2 Q12809 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP12 P39900 1/20 0.33
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
MMP16 P51512 1/20 0.33
MPO P05164 1/20 0.33
CASP1 P29466 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16316789 0.80 CYP3A4 (0.43) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL8993602 0.79 CYP3A4 (0.35) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL28748849 0.79 HTR2A (0.49) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL23270956 0.78 CYP3A4 (0.37) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6632884 0.78 CYP3A4 (0.37) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL27991976 0.74 LMNA (0.44) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL1106525 0.74 L3MBTL1 (0.52) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL26982399 0.74 CA1 (0.34) HTR2AHTR2CKCNH2L3MBTL1CASP1
SCHEMBL5618308 0.72 ESR1 (0.45) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL27718384 0.72 CYP3A4 (0.40) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104803956-A Synthesis method of firocoxib Jiangsu tianhe pharmaceutical co ltd 2015-07-29 CN claimed
CN-104803956-A Synthesis method of firocoxib Jiangsu tianhe pharmaceutical co ltd 2015-07-29 CN disclosed