SCHEMBL28019337

SCHEMBL28019337

C1=Nc2ccccc2CN1c1cccnc1

nearest known ligand 0.73

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.73
HPGD P15428 1/20 0.73
RAB9A P51151 1/20 0.73
SMN1; SMN2 Q16637 1/20 0.73
CYP11B2 P19099 3/20 0.46
NPSR1 Q6W5P4 1/20 0.41
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.38
CYP11B1 P15538 2/20 0.38
SIGMAR1 Q99720 1/20 0.37
CYP2A6 P11509 2/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2424631 0.87 NPC1 (0.96) NPC1HPGDRAB9ASMN1; SMN2NPSR1
SCHEMBL29417850 0.87 NPC1 (0.96) NPC1HPGDRAB9ASMN1; SMN2NPSR1
Formaldehyde SCHEMBL27861058 0.82 NPC1 (0.87) NPC1HPGDRAB9ASMN1; SMN2CYP11B2
SCHEMBL29546679 0.75 NPC1 (0.55) NPC1HPGDRAB9ASMN1; SMN2NPSR1
SCHEMBL7512518 0.74 NPC1 (0.67) NPC1HPGDRAB9ASMN1; SMN2NPSR1
SCHEMBL2428264 0.71 NPC1 (0.61) NPC1HPGDRAB9ASMN1; SMN2CYP11B2
SCHEMBL29547185 0.70 NPC1 (0.53) NPC1HPGDRAB9ASMN1; SMN2NPSR1
SCHEMBL2425683 0.65 RAB9A (0.57) NPC1HPGDRAB9ASMN1; SMN2CYP11B2
SCHEMBL904938 0.65 NPC1 (0.55) NPC1HPGDRAB9ASMN1; SMN2MEN1
SCHEMBL2013877 0.65 NPC1 (0.55) NPC1HPGDRAB9ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837832-B GDF-8 inhibitors 里格尔药品股份有限公司 2019-04-26 CN claimed
CN-104837832-A GDF-8 inhibitors RIGEL PHARMACEUTICALS INC 2015-08-12 CN claimed
CN-104837832-B GDF-8 inhibitors 里格尔药品股份有限公司 2019-04-26 CN disclosed
CN-106536507-A 2,3-disubstituted pyridine compounds as TGF-beta inhibitors and methods of use 里格尔药品股份有限公司 2017-03-22 CN disclosed
CN-104837832-A GDF-8 inhibitors RIGEL PHARMACEUTICALS INC 2015-08-12 CN disclosed