SCHEMBL28020311

SCHEMBL28020311

COCNC(=O)[CH]Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 8/20 0.41
HPGD P15428 5/20 0.41
CYP2C9 P11712 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CACNA1C Q13936 1/20 0.39
SCN9A Q15858 1/20 0.39
CA9 Q16790 1/20 0.39
CA13 Q8N1Q1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7749862 0.81 KMT2A (0.46) LMNAALDH1A1HPGDCYP2C9SMN1; SMN2
SCHEMBL4073041 0.79 ALDH1A1 (0.62) LMNAALDH1A1HPGDCYP2C9SMN1; SMN2
SCHEMBL294028 0.77 MAOB (0.43) LMNAKDM4EALDH1A1SMN1; SMN2CYP2C19
SCHEMBL6582849 0.77 MAOB (0.43) LMNAALDH1A1HPGDCYP2C9SMN1; SMN2
SCHEMBL27593026 0.77 KMT2A (0.57) LMNAKDM4EALDH1A1HPGDCYP2C9
SCHEMBL18343734 0.75 ALDH1A1 (0.46) LMNAALDH1A1HPGDCYP2C9SMN1; SMN2
SCHEMBL4324015 0.74 L3MBTL1 (0.59) LMNAALDH1A1HPGDSMN1; SMN2TDP1
SCHEMBL15229237 0.74 NPC1 (0.59) LMNAKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL4334225 0.73 ALDH1A1 (0.40) LMNAALDH1A1HPGDCYP2C9SMN1; SMN2
SCHEMBL7250131 0.73 KMT2A (0.63) ALDH1A1SMN1; SMN2MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854124-A Macrocyclic ketoamide immunoproteasome inhibitors HOFFMANN LA ROCHE 2015-08-19 CN disclosed