SCHEMBL28020837

SCHEMBL28020837

O=[N+]([O-])c1ccc2c(c1)CN(CCc1ccccc1)C2

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.58
KCNJ1 P48048 2/20 0.54
KCNH2 Q12809 1/20 0.54
HRH3 Q9Y5N1 1/20 0.51
GRIN2B Q13224 2/20 0.51
HTR2A P28223 2/20 0.50
PKM P14618 1/20 0.50
ABCB1 P08183 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6491669 0.90 ABCB1 (0.58) SIGMAR1KCNJ1KCNH2HRH3GRIN2B
SCHEMBL1997187 0.86 MAPT (0.50) SIGMAR1GRIN2BPKM
SCHEMBL6296037 0.78 DRD4 (0.54) SIGMAR1GRIN2BPKM
SCHEMBL6291722 0.78 GRIN2B (0.55) GRIN2BPKM
SCHEMBL21412716 0.78 HRH3 (0.55) SIGMAR1KCNJ1KCNH2HRH3GRIN2B
Hydrochloric Acid SCHEMBL8186681 0.77 GRIN2B (0.54) SIGMAR1GRIN2BPKM
SCHEMBL14067367 0.77 DPP7 (0.51) GRIN2B
SCHEMBL29383310 0.77 DPP7 (0.43) KCNJ1KCNH2GRIN2B
SCHEMBL7598211 0.77 ABCB1 (0.74) SIGMAR1KCNJ1KCNH2HRH3ABCB1
SCHEMBL1585063 0.77 SLC6A3 (0.61) SIGMAR1KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104744461-A Lactam-containing compounds and derivatives thereof as factor Xa inhibitors BRISTOL MYERS SQUIBB CO 2015-07-01 CN disclosed