SCHEMBL28021139

SCHEMBL28021139

Clc1c(-c2cccnc2)n[nH]c1-c1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.54
LRRK2 Q5S007 1/20 0.54
PIM1 P11309 3/20 0.49
MAP2K4 P45985 1/20 0.49
AXL P30530 1/20 0.48
CYP2A6 P11509 5/20 0.47
ALDH1A1 P00352 3/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
TTK P33981 1/20 0.44
CHEK1 O14757 1/20 0.44
BTK Q06187 1/20 0.44
CYP2E1 P05181 1/20 0.43
CYP2B6 P20813 1/20 0.43
PIM3 Q86V86 1/20 0.43
PIM2 Q9P1W9 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALK Q9UM73 1/20 0.42
METAP2 P50579 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15660759 0.93 IDO1 (0.55) IDO1LRRK2PIM1MAP2K4AXL
SCHEMBL3464003 0.81 MAP2K4 (0.55) IDO1LRRK2PIM1MAP2K4AXL
SCHEMBL16200084 0.78 CYP2A6 (0.41) IDO1LRRK2PIM1CYP2A6ALDH1A1
SCHEMBL13739801 0.76 ALDH1A1 (0.60) IDO1ALDH1A1CYP1A2CYP3A4TTK
SCHEMBL25288258 0.72 IDO1 (0.58) IDO1LRRK2PIM1MAP2K4AXL
SCHEMBL17279845 0.71 ALDH1A1 (0.50) IDO1MAP2K4ALDH1A1CYP1A2CYP3A4
SCHEMBL16670756 0.71 CYP2A6 (0.42) IDO1LRRK2PIM1MAP2K4CYP2A6
SCHEMBL22801811 0.71 FYN (0.43) IDO1LRRK2PIM1CYP2A6ALDH1A1
SCHEMBL22819372 0.71 IDO1 (0.60) IDO1LRRK2PIM1MAP2K4AXL
SCHEMBL9394628 0.70 IDO1 (0.56) IDO1LRRK2PIM1MAP2K4AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104860927-A 1H-3,5-bis(3-pyridinyl)-4-chloropyrazole compound, and preparation method and application thereof UNIV NINGBO 2015-08-26 CN claimed
CN-104860927-A 1H-3,5-bis(3-pyridinyl)-4-chloropyrazole compound, and preparation method and application thereof UNIV NINGBO 2015-08-26 CN disclosed
CN-104860927-A 1H-3,5-bis(3-pyridinyl)-4-chloropyrazole compound, and preparation method and application thereof UNIV NINGBO 2015-08-26 CN disclosed
CN-104860927-A 1H-3,5-bis(3-pyridinyl)-4-chloropyrazole compound, and preparation method and application thereof UNIV NINGBO 2015-08-26 CN disclosed