SCHEMBL28021722

SCHEMBL28021722

CCOC(=O)c1cc[c]s1.[Zn]

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
TSHR P16473 1/20 0.44
CA12 O43570 6/20 0.42
CA1 P00915 6/20 0.42
CA2 P00918 6/20 0.42
CA7 P43166 6/20 0.42
CA9 Q16790 6/20 0.42
CA14 Q9ULX7 6/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
CDC7 O00311 1/20 0.41
DBF4 Q9UBU7 1/20 0.41
CYP1A2 P05177 2/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAOA P21397 1/20 0.41
ALDH1A1 P00352 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL127564 0.98 HDAC3 (0.46) HDAC3HDAC4HDAC1HDAC6TSHR
SCHEMBL27769920 0.92 HDAC3 (0.42) HDAC3HDAC4HDAC1HDAC6TSHR
SCHEMBL127177 0.84 ALDH1A1 (0.49) TSHRESR1CYP1A2LMNACYP3A4
SCHEMBL10471051 0.84 ALDH1A1 (0.47) TSHRCDC7DBF4LMNAALDH1A1
SCHEMBL128695 0.81 TSHR (0.51) TSHRESR1CYP1A2LMNACYP3A4
SCHEMBL1641179 0.76 DGAT1 (0.38) HDAC3HDAC4HDAC1HDAC6
SCHEMBL4196673 0.73
SCHEMBL132083 0.73 CA12 (0.43) CA12CA1CA2CA7CA9
SCHEMBL7018973 0.72 HDAC3 (0.73) HDAC3HDAC4HDAC1HDAC6TSHR
SCHEMBL290059 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104876921-A 5H-cyclopenta[d]pyrimidines As AKT Protein Kinase Inhibitors ARRAY BIOPHARMA INC 2015-09-02 CN disclosed