SCHEMBL28021741

SCHEMBL28021741

O=C(O)Cc1c[nH]c(Cc2ccc([N+](=O)[O-])cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.43
PLA2G2A P14555 1/20 0.43
POLB P06746 1/20 0.43
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 2/20 0.42
GSK3B P49841 1/20 0.41
RIPK1 Q13546 1/20 0.41
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 2/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
ADORA2A P29274 1/20 0.39
TSHR P16473 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28021727 0.81 HRH3 (0.40) POLBCYP2C19CYP1A2RAB9AALDH1A1
SCHEMBL17154340 0.75 CYP2C19 (0.58) LTA4HPLA2G2APOLBCYP2C19CYP1A2
SCHEMBL28021740 0.74 ADORA2A (0.42) POLBCYP2C19CYP1A2RIPK1RAB9A
SCHEMBL16669003 0.74 MEN1 (0.43) POLBRAB9AMEN1KMT2AMAPT
SCHEMBL10587244 0.74 POLB (0.43) POLBCYP2C19CYP1A2GSK3BRIPK1
SCHEMBL22275961 0.73 CYP1B1 (0.39) CYP1A2GSK3BRAB9AALDH1A1KDM4E
SCHEMBL76204 0.73 CYP2C19 (0.64) CYP2C19CYP1A2ALDH1A1MEN1KMT2A
SCHEMBL30643815 0.73 CYP2C19 (0.64) CYP2C19CYP1A2ALDH1A1MEN1KMT2A
SCHEMBL1369959 0.71 CYP2C19 (0.62) CYP2C19CYP1A2ALDH1A1MEN1KMT2A
SCHEMBL27861234 0.71 CYP2C19 (0.62) CYP2C19CYP1A2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104768932-A Heteroaryl inhibitors of PDE4 TETRA DISCOVERY PARTNERS LLC 2015-07-08 CN disclosed