SCHEMBL10587244

SCHEMBL10587244

O=C(O)Cc1cnc(Cc2ccc([N+](=O)[O-])cc2)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.43
TSHR P16473 1/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 2/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
GSK3B P49841 1/20 0.41
RIPK1 Q13546 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8185024 0.85 TSHR (0.49) POLBTSHRMAPTALDH1A1CYP2C19
SCHEMBL7345076 0.82 BRS3 (0.49)
SCHEMBL6412219 0.77 POLB (0.50) POLBTSHRMAPTALDH1A1RIPK1
SCHEMBL7842828 0.77 BRS3 (0.54) PTGDR2GRIN1GRIN2B
SCHEMBL7039342 0.75 POLB (0.47) POLBTSHRMAPTALDH1A1RIPK1
SCHEMBL17154340 0.75 CYP2C19 (0.58) POLBTSHRMAPTALDH1A1CYP2C19
SCHEMBL28021741 0.74 LTA4H (0.43) POLBTSHRMAPTALDH1A1CYP2C19
SCHEMBL30643815 0.73 CYP2C19 (0.64) TSHRMAPTALDH1A1CYP2C19CYP1A2
SCHEMBL76204 0.73 CYP2C19 (0.64) TSHRMAPTALDH1A1CYP2C19CYP1A2
Hydrochloric Acid SCHEMBL8388746 0.73 CYP1A2 (0.46) CYP1A2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0324377-A2 Angiotensin II receptor blocking imidazoles and combinations thereof with diuretics and NSaids E.I. DU PONT DE NEMOURS AND COMPANY (US) 1989-07-19 EP disclosed