SCHEMBL28021740

SCHEMBL28021740

CC(=O)Oc1c[nH]c(Cc2ccc([N+](=O)[O-])cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.42
POLB P06746 1/20 0.41
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAOB P27338 1/20 0.40
RAB9A P51151 2/20 0.39
CCR5 P51681 1/20 0.39
GAA P10253 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPT P10636 1/20 0.38
RIPK1 Q13546 1/20 0.38
LMNA P02545 1/20 0.38
BCL9 O00512 1/20 0.37
CTNNB1 P35222 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28021725 0.82 ADORA2A (0.38) ADORA2APOLBGRIN1GRIN2BCYP1A2
SCHEMBL16669003 0.78 MEN1 (0.43) ADORA2APOLBRAB9AGAAMAPT
SCHEMBL28021741 0.74 LTA4H (0.43) ADORA2APOLBGRIN1GRIN2BCYP1A2
SCHEMBL2791412 0.71 CYP2C19 (0.43) POLBCYP1A2CYP2C9CYP2C19MAOB
SCHEMBL27758389 0.70 LMNA (0.36) RAB9ALMNA
SCHEMBL6016810 0.69 GAA (0.41) POLBCYP1A2CYP2C9CYP2C19MAOB
SCHEMBL5959134 0.68 MAOB (0.41) POLBCYP1A2CYP2C9CYP2C19MAOB
SCHEMBL5959150 0.68 MAOB (0.40) POLBCYP1A2CYP2C9CYP2C19MAOB
SCHEMBL27933983 0.67 GPR84 (0.35) MAPT
4-Nitrophenyl Acetate SCHEMBL74985 0.66 GAA (0.66) POLBMAOBGAAMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104768932-A Heteroaryl inhibitors of PDE4 TETRA DISCOVERY PARTNERS LLC 2015-07-08 CN disclosed