SCHEMBL28022103

SCHEMBL28022103

CCCCc1ccc2cnccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.42
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE10A Q9Y233 4/20 0.36
GSK3B P49841 1/20 0.36
LATS1 O95835 1/20 0.36
LATS2 Q9NRM7 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
TRPV1 Q8NER1 2/20 0.35
LTB4R Q15722 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
GPBAR1 Q8TDU6 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
CASP3 P42574 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10271357 0.82 HDAC1 (0.36) PDE10AHDAC3HDAC1HDAC2
SCHEMBL14911919 0.80 PDE10A (0.38) PDE10ALATS1LATS2HDAC3HDAC1
SCHEMBL538491 0.77 GPBAR1 (0.54) KCNH2PDE10AGPBAR1CYSLTR2CYSLTR1
Bromide SCHEMBL27600369 0.75 GPBAR1 (0.52) KCNH2PDE10AGPBAR1ALDH1A1MEN1
Hydrochloric Acid SCHEMBL27600363 0.75 GPBAR1 (0.52) KCNH2PDE10AGPBAR1ALDH1A1MEN1
SCHEMBL23554874 0.74 CCR1 (0.48) PDE10ALATS1LATS2HDAC3HDAC1
SCHEMBL29550107 0.74 CCR1 (0.48) PDE10ALATS1LATS2HDAC3HDAC1
SCHEMBL1161576 0.74 PDE3B (0.36) PDE10AHDAC3HDAC1HDAC2ALDH1A1
SCHEMBL10910525 0.74 GPBAR1 (0.51) KCNH2PDE10AGPBAR1ALDH1A1MEN1
SCHEMBL7512301 0.73 CCNC (0.44) CYSLTR2CYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104870459-B Metal complex 默克专利有限公司 2018-06-26 CN disclosed
CN-104870459-A Metal complexes MERCK PATENT GMBH 2015-08-26 CN disclosed
CN-104870458-A Metal complexes MERCK PATENT GMBH 2015-08-26 CN disclosed