SCHEMBL28022158

SCHEMBL28022158

[CH2]/C=C/c1ccc(Cl)cc1.[H+]

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.52
CYP1A2 P05177 2/20 0.48
HSD17B10 Q99714 2/20 0.46
FBP1 P09467 1/20 0.45
LMNA P02545 1/20 0.42
CYP2A6 P11509 1/20 0.42
ALOX5 P09917 1/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
NFE2L2 Q16236 1/20 0.42
MAOB P27338 2/20 0.41
HDAC2 Q92769 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL74363 0.97 AHR (0.54) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL74364 0.97 AHR (0.54) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL29190657 0.80 HDAC3 (0.50) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL699666 0.80 AHR (0.74) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL1795502 0.80 AHR (0.74) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL9679429 0.80 AHR (0.74) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL20582895 0.80 AHR (0.74) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL260347 0.80 AHR (0.74) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL9679426 0.80 AHR (0.74) AHRCYP1A2HSD17B10FBP1LMNA
SCHEMBL10458457 0.80 AHR (0.74) AHRCYP1A2HSD17B10FBP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104768932-B The heteroaryl inhibitors of PDE4 泰特拉探索合伙有限责任公司 2018-08-07 CN disclosed
CN-104768932-A Heteroaryl inhibitors of PDE4 TETRA DISCOVERY PARTNERS LLC 2015-07-08 CN disclosed