SCHEMBL28022277

SCHEMBL28022277

COC(=O)C(CO)NC(=O)C=Cc1ccccc1F

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 13/20 0.57
NOS3 P29474 9/20 0.57
NOS1 P29475 9/20 0.57
PTPN2 P17706 1/20 0.48
PTPN1 P18031 1/20 0.48
PTPN6 P29350 1/20 0.48
CDC25B P30305 1/20 0.48
MAOB P27338 1/20 0.46
TAS1R3 Q7RTX0 2/20 0.46
TAS1R1 Q7RTX1 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1711216 1.00 NOS2 (0.57) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL1711214 1.00 NOS2 (0.57) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL2194273 0.88 NOS2 (0.74) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL2194274 0.88 NOS2 (0.74) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL2194276 0.88 NOS2 (0.74) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL1710952 0.85 PTPN2 (0.55) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL1710949 0.85 PTPN2 (0.55) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL28820831 0.84 CYP3A4 (0.58) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL2190277 0.84 CYP3A4 (0.58) NOS2NOS3NOS1PTPN2PTPN1
SCHEMBL2190274 0.84 CYP3A4 (0.58) NOS2NOS3NOS1PTPN2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102216260-B Amino acid derivative NIPPON ZOKI PHARMACEUTICAL CO 2015-07-15 CN disclosed