SCHEMBL28022280

SCHEMBL28022280

O=C(O)c1cc2c(c(F)c1F)OCCC2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.44
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CTNNB1 P35222 2/20 0.36
WNT3A P56704 2/20 0.36
NOTUM Q6P988 1/20 0.35
XDH P47989 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
NPC1 O15118 1/20 0.34
MAP2K1 Q02750 2/20 0.33
MAPT P10636 1/20 0.33
GRM1 Q13255 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
HTR1A P08908 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29669545 0.92 PARP1 (0.53) PARP1ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL8481275 0.82 PARP1 (0.62) PARP1ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL25166008 0.78 PARP1 (0.49) PARP1ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL1142943 0.77 PARP1 (0.37) PARP1ALDH1A1KDM4ECTNNB1WNT3A
SCHEMBL7335337 0.75 HTR3A (0.43) PARP1ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL7395597 0.75 PARP1 (0.40) PARP1ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL9867616 0.75 PARP1 (0.40) PARP1ALDH1A1SMN1; SMN2KDM4EHPGD
Hydrochloric Acid SCHEMBL11514098 0.74 HTR3A (0.43) PARP1ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL14824890 0.74 PARP1 (0.33) PARP1CTNNB1WNT3ANOTUMHTR1A
SCHEMBL28022679 0.73 PARP1 (0.34) PARP1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104774188-A Benzohetercyclic or benzoheteraromatic-cyclic derivative and preparation method and application thereof in medicines JIANGSU HENGRUI MEDICINE CO 2015-07-15 CN disclosed