SCHEMBL28022368

SCHEMBL28022368

N#Cc1cccc(-c2ccccc2Cl)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.59
CYP2A6 P11509 1/20 0.52
AR P10275 1/20 0.50
KCNA5 P22460 1/20 0.50
KCNH2 Q12809 1/20 0.50
CLK4 Q9HAZ1 1/20 0.49
STK10 O94804 1/20 0.48
SLK Q9H2G2 1/20 0.48
MAOB P27338 1/20 0.47
ENPP1 P22413 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.45
GABRG2 P18507 2/20 0.44
GABRB3 P28472 2/20 0.44
GABRA5 P31644 2/20 0.44
GABRA3 P34903 2/20 0.44
PDK2 Q15119 1/20 0.44
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL996127 0.86 ADRA2C (0.64) ADRA2CCLK4MAOBGABRG2GABRB3
SCHEMBL10094705 0.84 ADRA2C (0.48) ADRA2CARKCNA5KCNH2CLK4
SCHEMBL31462934 0.84 ENPP1 (0.51) ADRA2CKCNA5KCNH2CLK4STK10
SCHEMBL11305092 0.83 CYP2A6 (0.54) ADRA2CCYP2A6ARMAOBGABRA5
SCHEMBL3422474 0.82 ADRA2C (0.60) ADRA2CCLK4MAOBGABRG2GABRB3
SCHEMBL31272452 0.82 ADRA2C (0.60) ADRA2CCLK4MAOBGABRG2GABRB3
SCHEMBL5217572 0.81 CYP2A6 (0.52) ADRA2CCYP2A6ARPDK2
SCHEMBL26272700 0.81 ADRA2C (0.48) ADRA2CCYP2A6KCNA5KCNH2CLK4
SCHEMBL23624364 0.80 ADRA2C (0.51) ADRA2CKCNA5KCNH2CLK4STK10
SCHEMBL10094533 0.80 KCNA5 (0.47) ADRA2CKCNA5KCNH2CLK4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108863850-A Biaryl base class compound and its preparation method and application 复旦大学 2018-11-23 CN disclosed
CN-105102449-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-25 CN disclosed