SCHEMBL28022537

SCHEMBL28022537

CC(C)(C)NC(=O)OCC1CN(c2ccc(C(F)(F)F)cc2)CCO1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.49
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
NOTUM Q6P988 1/20 0.42
SYK P43405 1/20 0.42
AKR1C3 P42330 1/20 0.40
DRD4 P21917 2/20 0.39
MDM2 Q00987 1/20 0.39
DRD2 P14416 1/20 0.38
PPARD Q03181 3/20 0.37
PPARA Q07869 3/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CA12 O43570 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CNR2 P34972 2/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28820861 0.82 NOTUM (0.50) TRPA1MAPTNOTUMDRD4DRD2
SCHEMBL27796251 0.79 SLC6A9 (0.46) TRPA1LMNAMAPTNOTUMAKR1C3
SCHEMBL15728297 0.79 TRPA1 (0.57) TRPA1LMNAMAPTNOTUMAKR1C3
SCHEMBL15719387 0.76 TRPA1 (0.60) TRPA1LMNAMAPTNOTUMAKR1C3
SCHEMBL28022536 0.74 TRPA1 (0.46) TRPA1LMNAMAPTNOTUMAKR1C3
SCHEMBL28597269 0.73 NOTUM (0.53) NOTUMDRD4DRD2CA12CA2
SCHEMBL22499928 0.73 NOTUM (0.53) NOTUMDRD4DRD2CA12CA2
SCHEMBL15728268 0.73 TRPA1 (0.47) TRPA1LMNAMAPTNOTUMAKR1C3
SCHEMBL28091529 0.72 DRD4 (0.55) DRD4DRD2CYP2D6
Hydrochloric Acid SCHEMBL15719216 0.72 TRPA1 (0.46) TRPA1LMNAMAPTNOTUMAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104812740-A Novel acetamide derivatives as TRP channel antagonists HOFFMANN LA ROCHE 2015-07-29 CN disclosed