SCHEMBL28022779

SCHEMBL28022779

Cc1ccc(Sc2ccncc2[N+](=O)[O-])cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.54
MAPT P10636 5/20 0.53
ALDH1A1 P00352 4/20 0.53
IDO1 P14902 1/20 0.53
PDE7A Q13946 4/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
NPSR1 Q6W5P4 2/20 0.50
HTT P42858 2/20 0.50
PDE4B Q07343 1/20 0.50
PDE4D Q08499 1/20 0.50
PDE7B Q9NP56 1/20 0.50
ALOX12 P18054 1/20 0.50
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 2/20 0.47
MAPK1 P28482 1/20 0.46
POLB P06746 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
GFER P55789 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16702465 0.84 PDE7A (0.55) MAPTALDH1A1PDE7AMEN1KMT2A
SCHEMBL8881808 0.78 MAPT (0.58) LMNAMAPTALDH1A1IDO1PDE7A
SCHEMBL2959825 0.78 MAPT (0.71) LMNAMAPTALDH1A1IDO1PDE7A
SCHEMBL31354776 0.77 CA12 (0.46) MAPTALDH1A1PDE7AMEN1KMT2A
SCHEMBL1137534 0.77 ALDH1A1 (0.47) LMNAMAPTALDH1A1PDE7AMEN1
SCHEMBL16702240 0.74 GSTP1 (0.49) MAPTALDH1A1PDE7AMEN1KMT2A
SCHEMBL8757145 0.74 MAPT (0.45) LMNAMAPTALDH1A1PDE7AMEN1
SCHEMBL7228444 0.73 PDE7A (0.39) LMNAMAPTALDH1A1PDE7AMEN1
SCHEMBL7228251 0.73 CYP1A2 (0.41) LMNAMAPTALDH1A1PDE7AMEN1
SCHEMBL16702882 0.73 ALDH1A1 (0.46) MAPTALDH1A1PDE7AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102807574-B New pyridine sulphur nitrogen seven-membered ring derivative as antitumor drug, and its preparation method and application CHANGCHUN DISCOVERY SCIENCES, LTD. (CN) 2015-09-02 CN disclosed