SCHEMBL28024258

SCHEMBL28024258

CCOC(=O)C1=C(C)N=C(O)NC1c1ccc(OC)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
LMNA P02545 3/20 0.54
GAA P10253 2/20 0.54
KDM4E B2RXH2 2/20 0.54
HPGD P15428 1/20 0.54
HSD17B10 Q99714 1/20 0.54
HTT P42858 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.50
POLB P06746 1/20 0.49
TSHR P16473 1/20 0.49
THRB P10828 1/20 0.48
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28024297 0.88 CA1 (0.48) ALDH1A1LMNAGAAKDM4EHSD17B10
SCHEMBL28141831 0.86 CA12 (0.48) ALDH1A1LMNAGAAHSD17B10HTT
SCHEMBL28142637 0.86 MAPT (0.50) ALDH1A1LMNAGAAKDM4EHSD17B10
SCHEMBL27897208 0.86 DHFR (0.57) ALDH1A1LMNAGAAKDM4EHTT
SCHEMBL28142608 0.84 HTT (0.57) ALDH1A1LMNAGAAKDM4EHSD17B10
SCHEMBL28843674 0.84 TP53 (0.43) ALDH1A1LMNAGAAKDM4EHSD17B10
SCHEMBL28821082 0.78 HSD17B10 (0.48) ALDH1A1LMNAHPGDHSD17B10CYP3A4
SCHEMBL3392657 0.76 GAA (0.76) ALDH1A1LMNAGAAKDM4EHPGD
SCHEMBL19752718 0.76 GAA (0.76) ALDH1A1LMNAGAAKDM4EHPGD
SCHEMBL3168404 0.75 CA1 (0.79) ALDH1A1LMNAGAAKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106632071-A Preparation method of 3, 4-dihydropyrimidine-2-ketone derivative through high-efficient catalyzation of ethyl alcohol promoted titanocene dichloride 陕西师范大学 2017-05-10 CN disclosed
CN-102993103-B N1, N3-dialkyl group replaces 3,4-dihydro-pyrimidin-2 ketone derivatives and preparation method thereof HUNAN SCI-TECH UNIV. (CN) 2015-07-29 CN disclosed