SCHEMBL28024313

SCHEMBL28024313

COc1ccc(C(F)F)cc1C1CC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.42
KRAS P01116 2/20 0.41
SOS1 Q07889 2/20 0.41
HTR2C P28335 2/20 0.40
MMP13 P45452 1/20 0.39
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
TACR1 P25103 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ACHE P22303 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21145969 0.88 MMP13 (0.43) HIF1AHTR2CMMP13TACR1CA1
SCHEMBL24758006 0.85 HIF1A (0.41) HIF1AHTR2CCA1CA2ACHE
SCHEMBL16950303 0.85 HIF1A (0.41) HIF1AKRASSOS1HTR2CMMP13
SCHEMBL16957130 0.79 HTR2C (0.37) HIF1AHTR2CMMP13HTR2A
SCHEMBL15577039 0.79 HIF1A (0.42) HIF1AMMP13TACR1
SCHEMBL21231846 0.77 SLC6A2 (0.54) HTR2CHTR2A
SCHEMBL21495050 0.76 MMP13 (0.36) HIF1AHTR2CMMP13PDE4APDE4B
SCHEMBL16950664 0.76 PPARG (0.41) HIF1AHTR2CPDE4ACA1CA2
SCHEMBL10192357 0.74 HIF1A (0.42) HIF1AMMP13PDE4APDE4BPDE4C
SCHEMBL13395132 0.74 CYP2D6 (0.42) CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102574861-B Methylpyrrolopyrimidinecarboxamides TAKEDA GMBH (DE) 2015-08-05 CN disclosed