SCHEMBL21495050

SCHEMBL21495050

COc1ccc([C@H](Br)C=O)cc1C1CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.36
HTR2C P28335 2/20 0.36
HIF1A Q16665 1/20 0.35
GAA P10253 1/20 0.35
USP9X Q93008 1/20 0.34
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
HTT P42858 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
ACHE P22303 1/20 0.33
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349469 0.79 GAA (0.50) GAAALDH1A1TSHRCA1CA2
SCHEMBL21145969 0.78 MMP13 (0.43) MMP13HTR2CHIF1AALDH1A1CA1
SCHEMBL16415970 0.76 SLC6A2 (0.43) GAAALDH1A1TSHRACHE
SCHEMBL28024313 0.76 HIF1A (0.42) MMP13HTR2CHIF1ACA1CA2
SCHEMBL7361147 0.76 PDE4A (0.54) PDE4APDE4BPDE4CPDE4D
SCHEMBL16957130 0.76 HTR2C (0.37) MMP13HTR2CHIF1AUSP9XALDH1A1
SCHEMBL24758006 0.75 HIF1A (0.41) HTR2CHIF1APTGDR2CA1CA2
SCHEMBL21495012 0.75 ALDH1A1 (0.53) GAAALDH1A1TSHRMEN1KMT2A
SCHEMBL15974455 0.75 ALDH1A1 (0.53) GAAALDH1A1TSHRMEN1KMT2A
SCHEMBL20425124 0.75 LMNA (0.44) GAAALDH1A1TSHRHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019201865-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2019-10-24 WO disclosed