SCHEMBL28024469

SCHEMBL28024469

c1ccc(COc2ccc3c(n2)CCCC3)nc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.43
ALOX15 P16050 2/20 0.41
PKM P14618 1/20 0.41
YWHAG P61981 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALDH1A1 P00352 2/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GRM1 Q13255 2/20 0.38
GABRA1 P14867 2/20 0.38
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
GABRA5 P31644 2/20 0.38
GABRA3 P34903 2/20 0.38
GABRA2 P47869 2/20 0.38
SYK P43405 1/20 0.37
AURKB Q96GD4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9300761 0.81 GRM5 (0.46) GRM5PKMNPSR1ALDH1A1HRH4
SCHEMBL10314867 0.79 BRD4 (0.45) GRM5ALDH1A1KDM4ESMN1; SMN2
SCHEMBL16872109 0.76 ACHE (0.44) GRM5ALOX15PKMYWHAGNPSR1
SCHEMBL16872369 0.76 ACHE (0.47) ALOX15ALDH1A1BCHEACHEGABRA1
SCHEMBL16872118 0.75 ACHE (0.46) ALOX15ALDH1A1BCHEACHEGABRA1
SCHEMBL4173286 0.73 ADRA2A (0.46) KDM4ESMN1; SMN2
SCHEMBL16872128 0.73 ACHE (0.44) GRM5ALOX15ALDH1A1BCHEACHE
SCHEMBL16872155 0.73 PIK3CA (0.43) GRM5ALOX15BCHEACHEKDM4E
SCHEMBL16151971 0.72 GRM5 (0.61) GRM5GRM1GABRG2GABRB3GABRA5
SCHEMBL28621695 0.71 SYK (0.44) BCHEACHESYKAURKBINCENP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104755471-A Pyridine derivative and drug NIPPON SHINYAKU CO LTD 2015-07-01 CN disclosed