SCHEMBL28025811

SCHEMBL28025811

CC(Oc1cc[n+]([O-])cc1C1CCC1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.36
SLC6A9 P48067 3/20 0.36
CNR2 P34972 15/20 0.35
CNR1 P21554 2/20 0.34
PDE4A P27815 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15777319 1.00 KCNH2 (0.36) KCNH2SLC6A9CNR2CNR1PDE4A
SCHEMBL15776052 0.76 PTGDR2 (0.39) CNR2
SCHEMBL15776455 0.75 RORC (0.33) KCNH2SLC6A9
SCHEMBL28026359 0.75 RORC (0.33) KCNH2SLC6A9
SCHEMBL15777436 0.73 CNR2 (0.44) CNR2CNR1
SCHEMBL28026358 0.73 CNR2 (0.44) CNR2CNR1
SCHEMBL16115704 0.70 CNR2 (0.40) CNR2
SCHEMBL28026344 0.65 GPR84 (0.37) SLC6A9
SCHEMBL28026343 0.65 GPR84 (0.37) SLC6A9
SCHEMBL15777727 0.63 CNR2 (0.54) CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837818-A Pyridine-2-amides useful as CB2 agonists HOFFMANN LA ROCHE 2015-08-12 CN disclosed