SCHEMBL28025970

SCHEMBL28025970

COC(=O)N(c1cccc([N+](=O)[O-])c1)C(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 7/20 0.44
KMT2A Q03164 7/20 0.44
LMNA P02545 3/20 0.44
MAPT P10636 7/20 0.43
HTT P42858 2/20 0.43
TSHR P16473 1/20 0.43
DDX3X O00571 1/20 0.43
POLB P06746 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.43
MAPK1 P28482 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HSP90AA1 P07900 1/20 0.43
HPGD P15428 1/20 0.43
CACNA1B Q00975 1/20 0.43
APBA1 Q02410 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NLRP1 Q9C000 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2453168 0.84 TP53 (0.49) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL2453170 0.84 TP53 (0.49) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL1815772 0.80 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL2311749 0.80 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL2312487 0.80 MEN1 (0.48) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL4014610 0.78 ALDH1A1 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL1028316 0.77 OPRM1 (0.43) ALDH1A1MEN1KMT2AMAPTPOLB
SCHEMBL1027116 0.76 MAOB (0.47) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL1027117 0.76 MAOB (0.47) SMN1; SMN2ALDH1A1MEN1KMT2ALMNA
SCHEMBL18053692 0.76 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104755461-A 6-aminoindole derivatives as TRP channel antagonists HOFFMANN LA ROCHE 2015-07-01 CN disclosed