SCHEMBL28026029

SCHEMBL28026029

Cc1c(C(=O)O)cc(-c2ccc(Cl)cc2)cc1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 5/20 0.56
AKR1C1 Q04828 5/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
AURKA O14965 1/20 0.54
TPX2 Q9ULW0 1/20 0.54
FTO Q9C0B1 1/20 0.49
MCL1 Q07820 1/20 0.49
RXRA P19793 1/20 0.48
RXRB P28702 1/20 0.48
NOTUM Q6P988 2/20 0.47
ALAD P13716 1/20 0.47
TP53 P04637 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALDH1A1 P00352 2/20 0.47
TSHR P16473 1/20 0.47
CASP1 P29466 1/20 0.47
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10024251 0.83 MCL1 (0.54) AKR1C2AKR1C1NPC1RAB9AAURKA
SCHEMBL14018381 0.83 NPC1 (0.48) AKR1C2AKR1C1NPC1RAB9AAURKA
SCHEMBL27786187 0.82 PTPN1 (0.58) AKR1C2AKR1C1MCL1ALDH1A1
SCHEMBL27808113 0.81 BCL2L1 (0.53) AKR1C2AKR1C1MCL1RXRARXRB
SCHEMBL28201908 0.81 RXFP1 (0.51) AKR1C2AKR1C1MCL1RXRARXRB
SCHEMBL28201890 0.81 TDP1 (0.53) AKR1C2AKR1C1MCL1RXRARXRB
SCHEMBL10024263 0.79 RXRB (0.58) AKR1C2AKR1C1NPC1RAB9AMCL1
SCHEMBL13537088 0.79 AKR1C4 (0.56) AKR1C2AKR1C1NPC1RAB9AAURKA
SCHEMBL28840070 0.79 ALDH1A1 (0.55) AKR1C2AKR1C1AURKATPX2NOTUM
SCHEMBL11064733 0.78 MAP4K4 (0.50) AKR1C2AKR1C1NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105473568-A 1, 7-naphthyridine derivatives HOFFMANN LA ROCHE 2016-04-06 CN claimed
CN-104755473-B 2,3 benzodiazepine * 拜耳医药股份有限公司 2017-03-08 CN disclosed
CN-105473568-A 1, 7-naphthyridine derivatives HOFFMANN LA ROCHE 2016-04-06 CN disclosed
CN-104755473-A 2,3-benzodiazepines Bayer Pharma AG 2015-07-01 CN disclosed