SCHEMBL28026341

SCHEMBL28026341

C[C@H](Oc1ccc(C#N)nc1)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.40
S1PR1 P21453 1/20 0.35
DGAT1 O75907 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
CHEK1 O14757 3/20 0.34
ACACB O00763 2/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
AR P10275 2/20 0.33
CTSS P25774 1/20 0.32
NR3C1 P04150 1/20 0.32
CNR2 P34972 1/20 0.32
PIK3CD O00329 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
HCK P08631 1/20 0.32
SRC P12931 1/20 0.32
KDR P35968 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506514 1.00 TRPA1 (0.40) TRPA1S1PR1DGAT1SCN10ACHEK1
SCHEMBL10229621 0.88 TRPA1 (0.36) TRPA1S1PR1DGAT1SCN10ACHEK1
SCHEMBL12923711 0.81 ACACB (0.44) SCN10AACACBALOX5APFEN1PIK3CD
SCHEMBL2335107 0.78 KDR (0.41) ACACBALOX5APFEN1CTSSKDR
SCHEMBL19614572 0.76 GAA (0.44) TRPA1NR3C1
SCHEMBL19614569 0.76 GAA (0.44) TRPA1NR3C1
SCHEMBL250730 0.76 GAA (0.44) TRPA1NR3C1
SCHEMBL22397178 0.75 TRPA1 (0.43) TRPA1DGAT1CHEK1ALOX5APFEN1
SCHEMBL29078782 0.75 ALOX5AP (0.37) TRPA1CHEK1ALOX5APFEN1NSD2
SCHEMBL29620884 0.74 TRPA1 (0.55) TRPA1DGAT1SCN10AALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837818-A Pyridine-2-amides useful as CB2 agonists HOFFMANN LA ROCHE 2015-08-12 CN disclosed