SCHEMBL28026367

SCHEMBL28026367

C[C@H](Oc1cccnc1)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.46
CHRNA4 P43681 7/20 0.46
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
CYP3A4 P08684 2/20 0.43
CYP3A5 P20815 2/20 0.43
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HTT P42858 1/20 0.39
GRM2 Q14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28026369 1.00 CHRNB2 (0.46) CHRNB2CHRNA4CHRNB4CHRNA3CYP3A4
SCHEMBL11911979 0.84 CHRNB2 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3CYP3A4
SCHEMBL4946642 0.79 CHRNB2 (0.51) CHRNB2CHRNA4CHRNB4CHRNA3CYP3A4
SCHEMBL29854164 0.79 CHRNB2 (0.51) CHRNB2CHRNA4CHRNB4CHRNA3CYP3A4
SCHEMBL30361331 0.77 CYP3A4 (0.38) CYP3A4CYP3A5LMNATDP1
SCHEMBL18833426 0.77 KDM4E (0.39) CHRNB4CHRNA3LMNA
SCHEMBL28060320 0.77 KDM4E (0.39) CHRNB4CHRNA3LMNA
Trifluoroacetic Acid SCHEMBL30901022 0.76 CYP3A4 (0.51) CHRNB2CHRNA4CHRNB4CHRNA3CYP3A4
SCHEMBL14477064 0.76 CHRNB2 (0.49) CHRNB2CHRNA4CHRNB4CHRNA3CYP3A4
SCHEMBL1515202 0.76 CHRNB2 (0.49) CHRNB2CHRNA4CHRNB4CHRNA3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837818-A Pyridine-2-amides useful as CB2 agonists HOFFMANN LA ROCHE 2015-08-12 CN disclosed