SCHEMBL28027249

SCHEMBL28027249

Cc1c(-c2cccc(CN)c2)nc2ccccc2c1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
TLR8 Q9NR97 2/20 0.43
TSHR P16473 1/20 0.43
PDE10A Q9Y233 1/20 0.43
DHODH Q02127 1/20 0.41
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28027282 0.89 DHODH (0.49) TLR8TSHRPDE10ADHODHSMN1; SMN2
SCHEMBL28159697 0.81 KMT2A (0.50) TSHRPDE10ADHODHESR1ESR2
SCHEMBL27651468 0.81 ESR1 (0.51) NOS3NOS1NOS2TLR8ESR1
SCHEMBL13758058 0.81 PDE10A (0.60) TSHRPDE10ADHODHESR1ESR2
SCHEMBL28027245 0.79 PRNP (0.46) TSHRPDE10ADHODHESR1ESR2
SCHEMBL28027244 0.79 PTGS1 (0.54) TSHRPDE10ADHODHESR1ESR2
SCHEMBL28027246 0.77 DHODH (0.55) DHODH
SCHEMBL28159695 0.75 TDP1 (0.66) TSHRPDE10ADHODH
SCHEMBL27651467 0.73 TAAR1 (0.55) TLR8TSHRESR1ESR2SMN1; SMN2
SCHEMBL28159698 0.73 DHODH (0.52) TSHRPDE10ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104817496-B A kind of 1,2,3,4 tetrahydroquinoline derivatives and preparation method thereof 中国科学院化学研究所 2017-06-16 CN disclosed
CN-104817496-A 1, 2, 3, 4-tetrahydroquinoline derivative and method for preparing same CHINESE ACAD INST CHEMISTRY 2015-08-05 CN disclosed