SCHEMBL28027282

SCHEMBL28027282

Cc1c(-c2ccc(CN)cc2)nc2ccccc2c1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.49
PDE10A Q9Y233 2/20 0.48
TSHR P16473 1/20 0.48
TAAR1 Q96RJ0 1/20 0.47
TDP1 Q9NUW8 1/20 0.45
TOP1 P11387 1/20 0.44
LMNA P02545 1/20 0.42
ADORA2A P29274 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TLR8 Q9NR97 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28027249 0.89 NOS3 (0.45) DHODHPDE10ATSHRSMN1; SMN2TLR8
SCHEMBL13758058 0.86 PDE10A (0.60) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28027246 0.84 DHODH (0.55) DHODHTAAR1
SCHEMBL28159695 0.83 TDP1 (0.66) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL27651467 0.81 TAAR1 (0.55) TSHRTAAR1TDP1LMNASMN1; SMN2
SCHEMBL28027827 0.81 ADORA2A (0.53) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28027826 0.81 KDM4E (0.62) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28027828 0.81 KDM4E (0.62) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28159698 0.81 DHODH (0.52) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL14119243 0.80 TAAR1 (0.63) TAAR1TDP1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104817496-B A kind of 1,2,3,4 tetrahydroquinoline derivatives and preparation method thereof 中国科学院化学研究所 2017-06-16 CN disclosed
CN-104817496-A 1, 2, 3, 4-tetrahydroquinoline derivative and method for preparing same CHINESE ACAD INST CHEMISTRY 2015-08-05 CN disclosed