SCHEMBL28159698

SCHEMBL28159698

Cc1c(-c2ccccc2)nc2ccccc2c1-c1ccc(Br)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.52
PDE10A Q9Y233 2/20 0.51
TSHR P16473 1/20 0.51
TDP1 Q9NUW8 1/20 0.49
TOP1 P11387 1/20 0.47
LMNA P02545 1/20 0.45
PRNP P04156 2/20 0.45
RXFP1 Q9HBX9 2/20 0.45
PPARG P37231 1/20 0.45
NR2E3 Q9Y5X4 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
CYP1A1 P04798 2/20 0.44
CYP1B1 Q16678 2/20 0.44
CYP1A2 P05177 1/20 0.44
ALDH1A1 P00352 1/20 0.44
AKR1B10 O60218 1/20 0.44
TNKS O95271 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13758058 0.90 PDE10A (0.60) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28159695 0.87 TDP1 (0.66) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL18804452 0.85 DHODH (0.45) DHODHPDE10ATSHRTDP1RXFP1
SCHEMBL28027245 0.85 PRNP (0.46) DHODHPDE10ATSHRLMNAPRNP
SCHEMBL28027828 0.84 KDM4E (0.62) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28027826 0.84 KDM4E (0.62) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28027827 0.84 ADORA2A (0.53) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL28160154 0.82 ALDH1A1 (0.67) DHODHPDE10ATSHRTDP1LMNA
SCHEMBL28027282 0.81 DHODH (0.49) DHODHPDE10ATSHRTDP1TOP1
SCHEMBL29488292 0.79 ESR1 (0.56) TDP1RXFP1CYP1A1CYP1B1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104817496-B A kind of 1,2,3,4 tetrahydroquinoline derivatives and preparation method thereof 中国科学院化学研究所 2017-06-16 CN disclosed
CN-104817496-A 1, 2, 3, 4-tetrahydroquinoline derivative and method for preparing same CHINESE ACAD INST CHEMISTRY 2015-08-05 CN disclosed