SCHEMBL28028200

SCHEMBL28028200

O=C(O)CCC(F)(F)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
FFAR1 O14842 2/20 0.47
HDAC3 O15379 1/20 0.47
MAPK1 P28482 1/20 0.47
ADRA1A P35348 1/20 0.47
HDAC4 P56524 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
CES1 P23141 5/20 0.46
HIF1A Q16665 1/20 0.46
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15619550 0.89 SMN1; SMN2 (0.53) KEAP1SMN1; SMN2FFAR1HDAC3MAPK1
SCHEMBL2344852 0.85 SMN1; SMN2 (0.47) KEAP1SMN1; SMN2CES1HIF1ACYP2C19
SCHEMBL28044400 0.81 CA12 (0.49) FFAR1MAPK1PTPN1
SCHEMBL4138709 0.80 CES1 (0.48) KEAP1SMN1; SMN2FFAR1HDAC3MAPK1
SCHEMBL29633636 0.78 TDP1 (0.44) SMN1; SMN2CES1HIF1ACYP2C19FDPS
SCHEMBL21328934 0.78 ALDH1A1 (0.47) KEAP1FFAR1CES1
SCHEMBL5750633 0.77 KEAP1 (0.50) KEAP1SMN1; SMN2FFAR1HDAC3MAPK1
SCHEMBL7432415 0.77 SMN1; SMN2 (0.50) KEAP1SMN1; SMN2FFAR1HDAC3MAPK1
SCHEMBL19224281 0.76 SLC6A2 (0.50) SMN1; SMN2CES1HIF1ACYP2C19FDPS
SCHEMBL26748568 0.75 TAAR1 (0.41) SMN1; SMN2CES1HIF1ACYP2C19FDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102417480-B As the Spirocyclic nitriles of proteinase inhibitor Sanofi-Aventis S. P. A. (FR) 2015-08-26 CN disclosed