SCHEMBL28028586

SCHEMBL28028586

O=C(O)Cc1ncccc1OCC(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 3/20 0.46
CACNA1G O43497 2/20 0.46
SSTR4 P31391 3/20 0.42
MAPT P10636 2/20 0.41
CYP1A2 P05177 2/20 0.41
KDM4E B2RXH2 2/20 0.41
AGBL2 Q5U5Z8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CFD P00746 1/20 0.40
MEN1 O00255 1/20 0.40
S1PR2 O95136 1/20 0.40
S1PR4 O95977 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
XBP1 P17861 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
PAX8 Q06710 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30851832 0.81 ALDH1A1 (0.47) CACNA1HCACNA1GSSTR4MAPTCYP1A2
SCHEMBL27518122 0.80 KDM4E (0.44) MAPTCYP1A2KDM4EL3MBTL1CFD
SCHEMBL459180 0.78 MAPT (0.47) CACNA1HCACNA1GSSTR4MAPTCYP1A2
SCHEMBL4538802 0.78 TRPV1 (0.45) SSTR4MAPTCYP1A2KDM4EAGBL2
SCHEMBL24180073 0.78 SSTR4 (0.40) CACNA1HCACNA1GSSTR4MAPTCYP1A2
SCHEMBL29796455 0.78 SMN1; SMN2 (0.50) MAPTCYP1A2KDM4EMEN1LMNA
SCHEMBL7371029 0.78 MAPT (0.42) CACNA1HCACNA1GSSTR4MAPTCYP1A2
SCHEMBL30852196 0.78 CACNA1H (0.39) CACNA1HCACNA1GSSTR4MAPTCYP1A2
SCHEMBL16364773 0.78 SMN1; SMN2 (0.50) MAPTCYP1A2KDM4EMEN1LMNA
SCHEMBL22553411 0.77 MAPT (0.41) MAPTCYP1A2KDM4ECFDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958922-B 2,5,6,7-tetrahydrochysene-[Isosorbide-5-Nitrae] oxygen azepine *-3-base amine or 2,3,6,7-tetrahydrochysene-[Isosorbide-5-Nitrae] oxygen azepine *-5-ylamine compounds HOFFMAN-LA ROCHE LTD. (CH) 2015-09-30 CN disclosed