SCHEMBL28028898

SCHEMBL28028898

COc1ccccc1Cn1c(=O)[nH]c2c(N[C]=O)nc(-c3cc[nH]n3)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.46
NUDT1 P36639 1/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
PRNP P04156 2/20 0.38
ADORA2A P29274 3/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
TLR7 Q9NYK1 3/20 0.36
RXFP1 Q9HBX9 2/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HTR3A P46098 1/20 0.35
EPHX2 P34913 1/20 0.35
KDM1A O60341 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28028874 0.84 MTOR (0.47) MTORNUDT1MEN1KMT2APRNP
SCHEMBL28028882 0.84 MTOR (0.59) MTORNUDT1MEN1KMT2APRNP
SCHEMBL28821952 0.82 MTOR (0.47) MTORNUDT1MEN1KMT2APRNP
SCHEMBL28028878 0.81 MTOR (0.48) MTORMEN1KMT2AALDH1A1KDM4E
SCHEMBL28029238 0.81 MTOR (0.44) MTORNUDT1MEN1KMT2APRNP
SCHEMBL28028900 0.81 ADORA2A (0.46) MTORNUDT1MEN1KMT2APRNP
SCHEMBL28029224 0.81 MTOR (0.43) MTORNUDT1MEN1KMT2APRNP
SCHEMBL28029222 0.81 CYP1A2 (0.54) MTORMEN1KMT2AADORA2AADORA1
SCHEMBL28948857 0.79 GRIN1 (0.46) MTORMEN1KMT2AADORA2ALMNA
SCHEMBL28028876 0.79 MTOR (0.46) MTORNUDT1MEN1KMT2APRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107976546-A Inhibition of phosphorylation to TOR kinase inhibiting activities mark PRAS40, GSK3- β or P70S6K1 西格诺药品有限公司 2018-05-01 CN disclosed
CN-104870998-B inhibition of phosphorylation of PRAS40, GSK3- β or P70S6K1 as a marker of TOR kinase inhibitory activity 西格诺药品有限公司 2018-02-02 CN disclosed
CN-104870998-A Inhibition of phosphorylation of PRAS40, GSK 3-beta or P70S6K1 as a marker of TOR kinase inhibitory activity SIGNAL PHARM LLC 2015-08-26 CN disclosed