SCHEMBL28029029

SCHEMBL28029029

CC(C)(C)OC(=O)N1CCC(C(=O)O)(c2cccc(Br)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
ALOX15 P16050 1/20 0.52
ATM Q13315 1/20 0.52
TACR1 P25103 1/20 0.46
KMT2A Q03164 3/20 0.45
RORC P51449 2/20 0.45
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
JAK2 O60674 1/20 0.43
JAK1 P23458 1/20 0.43
USP30 Q70CQ3 2/20 0.43
TET3 O43151 1/20 0.42
FBXL19 Q6PCT2 1/20 0.42
CXXC5 Q7LFL8 1/20 0.42
TET1 Q8NFU7 1/20 0.42
KDM2B Q8NHM5 1/20 0.42
CXXC4 Q9H2H0 1/20 0.42
KDM2A Q9Y2K7 1/20 0.42
GPR119 Q8TDV5 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31694033 1.00 TSHR (0.52) TSHRALOX15ATMTACR1KMT2A
SCHEMBL30056366 0.93 TSHR (0.47) TSHRALOX15ATMTACR1KMT2A
SCHEMBL27167101 0.93 TSHR (0.47) TSHRALOX15ATMTACR1KMT2A
SCHEMBL19331220 0.89 TSHR (0.48) TSHRALOX15ATMTACR1KMT2A
SCHEMBL972474 0.86 TSHR (0.65) TSHRALOX15ATMTACR1KMT2A
SCHEMBL29135477 0.86 TSHR (0.45) TSHRALOX15ATMTACR1KMT2A
SCHEMBL30775694 0.86 TSHR (0.45) TSHRALOX15ATMTACR1KMT2A
SCHEMBL2577367 0.86 TSHR (0.52) TSHRALOX15ATMTACR1KMT2A
SCHEMBL19690249 0.85 TSHR (0.46) TSHRALOX15ATMTACR1KMT2A
SCHEMBL12988312 0.85 TSHR (0.53) TSHRALOX15ATMTACR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104876934-B A kind of nitrogen heterocyclic ring phenylpiperidine compound and preparation method and application 山东大学 2017-08-11 CN disclosed
CN-104876934-A Nitrogen-containing heterocyclic phenyl piperidine compound as well as preparation method and application thereof UNIV SHANDONG 2015-09-02 CN disclosed