SCHEMBL30056366

SCHEMBL30056366

CC(C)(C)OC(=O)N1CCC(C(=O)O)(c2cccc(Br)c2)C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
ALOX15 P16050 1/20 0.47
ATM Q13315 1/20 0.47
USP30 Q70CQ3 3/20 0.46
RORC P51449 4/20 0.46
SCD5 Q86SK9 1/20 0.43
TACR1 P25103 1/20 0.42
KMT2A Q03164 2/20 0.41
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
CYP11B2 P19099 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27167101 1.00 TSHR (0.47) TSHRALOX15ATMUSP30RORC
SCHEMBL28029029 0.93 TSHR (0.52) TSHRALOX15ATMUSP30RORC
SCHEMBL31694033 0.93 TSHR (0.52) TSHRALOX15ATMUSP30RORC
SCHEMBL30775694 0.91 TSHR (0.45) TSHRALOX15ATMUSP30RORC
SCHEMBL29135477 0.91 TSHR (0.45) TSHRALOX15ATMUSP30RORC
SCHEMBL21408986 0.87 TSHR (0.60) TSHRALOX15ATMUSP30RORC
SCHEMBL19183400 0.87 TSHR (0.60) TSHRALOX15ATMUSP30RORC
SCHEMBL19331220 0.85 TSHR (0.48) TSHRALOX15ATMUSP30RORC
SCHEMBL38652021 0.83 USP30 (0.49) TSHRALOX15ATMUSP30RORC
SCHEMBL19690249 0.81 TSHR (0.46) TSHRALOX15ATMUSP30RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4333982-A1 PKC-THETA MODULATORS Exscientia Al Limited (GB) 2024-03-13 EP disclosed
WO-2022234298-A1 PKC-THETA MODULATORS EXSCIENTIA AI LIMITED (GB) 2022-11-10 WO disclosed