SCHEMBL28029680

SCHEMBL28029680

O=Cc1nc2ccccc2o1.[H+]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54
HDAC11 Q96DB2 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HDAC9 Q9UKV0 1/20 0.54
HDAC5 Q9UQL6 1/20 0.54
SNCA P37840 1/20 0.50
ADAMTS5 Q9UNA0 1/20 0.48
MAPT P10636 5/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
TP53 P04637 3/20 0.47
LMNA P02545 2/20 0.47
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
MEN1 O00255 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL223564 0.98 HDAC3 (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
Quinoline SCHEMBL27330442 0.85 ALDH1A1 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6421501 0.81 SNCA (0.64) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6421503 0.81 SNCA (0.64) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7472170 0.79 SNCA (0.62) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7472176 0.79 SNCA (0.62) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8718548 0.79 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6607140 0.79 MEN1 (0.63) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6607138 0.79 MEN1 (0.63) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8718547 0.79 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476664-A New compound as autotaxin inhibitors and the pharmaceutical composition comprising it 乐高化学生物科学股份有限公司 2019-03-15 CN disclosed
CN-109121397-A Heterocyclic compound, especially 2- oxo -4,4,5,5,6,6,7,7- octahydro benzoxazoles derivatives and their purposes as antimicrobial compound 莱德克斯制药公共有限公司 2019-01-01 CN disclosed
CN-106749080-A The plant growth regulator and its preparation method and purposes of high resistance to cold and diseases 中国科学院上海生命科学研究院 2017-05-31 CN disclosed
CN-103842348-B Selective androgen receptor modulators ELI LILLY AND CO. (US) 2015-08-19 CN disclosed