SCHEMBL28030256

SCHEMBL28030256

CC(=O)Oc1cc([N+](=O)[O-])c(F)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
ITGB1 P05556 1/20 0.42
ITGA5 P08648 1/20 0.42
ATM Q13315 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ESPL1 Q14674 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 6/20 0.40
HIF1A Q16665 1/20 0.40
HTT P42858 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
HSPB1 P04792 2/20 0.38
MAPT P10636 3/20 0.38
VCAM1 P19320 1/20 0.38
VCP P55072 1/20 0.38
GAA P10253 3/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17375034 0.87 TTR (0.41) CYP4F2CYP4A11ITGB1ITGA5ATM
SCHEMBL28136377 0.87 ITGB1 (0.40) CYP4F2CYP4A11ITGB1ITGA5ATM
SCHEMBL10719888 0.87 SMN1; SMN2 (0.42) CYP4F2CYP4A11ITGB1ITGA5ATM
SCHEMBL17466056 0.86 LMNA (0.40) CYP4F2CYP4A11ITGB1ITGA5ATM
SCHEMBL7215856 0.84 HTT (0.41) ATMTDP1ESPL1SMN1; SMN2ALDH1A1
SCHEMBL16513277 0.83 ATM (0.41) ITGB1ITGA5ATMTDP1ESPL1
SCHEMBL23850947 0.83 ALDH1A1 (0.44) TDP1SMN1; SMN2ALDH1A1HTTLMNA
SCHEMBL810412 0.80 ALDH1A1 (0.43) TDP1ESPL1SMN1; SMN2ALDH1A1MEN1
SCHEMBL512256 0.79 ALDH1A1 (0.51) ATMTDP1ESPL1ALDH1A1HIF1A
SCHEMBL29804996 0.79 ALDH1A1 (0.51) ATMTDP1ESPL1ALDH1A1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026052-B 5-hydroxyalkyl benzimidazoles as mIDH1 inhibitors 德国癌症研究公共权益基金会 2021-10-08 CN disclosed
CN-107810176-B N-menthyl benzimidazoles as mIDH1 inhibitors 德国癌症研究公共权益基金会 2020-10-16 CN disclosed
CN-110433162-A It can be used as the dihydronaphthridine and related compound of the kinase inhibitor for treating proliferative disease DECIPHERA PHARMACEUTICALS LLC 2019-11-12 CN disclosed
CN-110403938-A It can be used as the dihydronaphthridine and related compound of the kinase inhibitor for treating proliferative disease DECIPHERA PHARMACEUTICALS LLC 2019-11-05 CN disclosed
CN-104902895-B Dihydronaphthyridines and related compounds useful as kinase inhibitors for the treatment of proliferative diseases 德西费拉制药有限责任公司 2019-03-29 CN disclosed
CN-104902895-A Dihydronaphthyridines and related compounds useful as kinase inhibitors for the treatment of proliferative diseases FLYNN DANIEL L 2015-09-09 CN disclosed