SCHEMBL28030276

SCHEMBL28030276

COc1ccc2cc(C(Cl)c3ccccc3)ccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.41
KDM4E B2RXH2 2/20 0.38
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CDK6 Q00534 1/20 0.35
ALDH1A1 P00352 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HPGD P15428 2/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
SLC6A3 Q01959 4/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2D6 P10635 3/20 0.34
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 3/20 0.34
KCNH2 Q12809 3/20 0.34
BCL2L11 O43521 1/20 0.34
BID P55957 1/20 0.34
BCL2L1 Q07817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14288343 0.78 CDK4 (0.41) KDM4ECDK4CCND1CDK6ALDH1A1
SCHEMBL20666274 0.75 CDK4 (0.37) ADORA1KDM4ECDK4CCND1CDK6
SCHEMBL11832003 0.75 UGT2B7 (0.49) KDM4ECDK4CCND1CDK6HPGD
SCHEMBL21164372 0.74 BCL2L11 (0.40) ADORA1KDM4ECDK4CCND1CDK6
SCHEMBL11827253 0.73 AKR1C3 (0.61) AKR1C3AKR1C2
SCHEMBL12695592 0.73 BACE1 (0.57) ADORA1KDM4EALDH1A1NPC1RAB9A
SCHEMBL23848110 0.73 ABCB11 (0.43) CDK4CCND1CDK6ALDH1A1HPGD
SCHEMBL11839847 0.72 AKR1C3 (0.37) ADORA1KDM4ECDK4CCND1CDK6
SCHEMBL4574921 0.71 SLC6A2 (0.51) KMT2ASLC6A3CYP3A4CYP2D6SLC6A2
Benzene SCHEMBL27589371 0.71 KDM4E (0.52) KDM4EALDH1A1NPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103242231-B Quinoline derivatives and preparation method thereof and application TIANJIN GREENPINE PHARMA CO., LTD. (CN) 2015-10-28 CN disclosed