SCHEMBL28030655

SCHEMBL28030655

NC(=O)Cc1cccc(N2CCCC2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.58
ITGB3 P05106 2/20 0.56
ITGA2B P08514 2/20 0.56
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 3/20 0.55
MEN1 O00255 2/20 0.55
HPGD P15428 2/20 0.55
KMT2A Q03164 2/20 0.55
MAPT P10636 2/20 0.55
POLB P06746 2/20 0.55
USP2 O75604 1/20 0.55
BLM P54132 1/20 0.55
KCNQ2 O43526 2/20 0.53
GAA P10253 1/20 0.53
HSD17B10 Q99714 1/20 0.53
PRMT6 Q96LA8 1/20 0.53
CNR1 P21554 1/20 0.47
KLKB1 P03952 1/20 0.46
KLK1 P06870 1/20 0.46
HTR1A P08908 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29639816 0.98 AGXT (0.56) AGXTITGB3ITGA2BKDM4EALDH1A1
SCHEMBL20392367 0.97 ITGB3 (0.56) AGXTITGB3ITGA2BKDM4EALDH1A1
SCHEMBL5177552 0.86 AGXT (0.61) AGXTITGB3ITGA2BMEN1KMT2A
SCHEMBL5790195 0.86 AGXT (0.61) AGXTITGB3ITGA2BHTR1AHTR2A
SCHEMBL17115677 0.84 AGXT (0.58) AGXTITGB3ITGA2BKDM4EALDH1A1
SCHEMBL16880373 0.82 ITGB3 (0.64) AGXTITGB3ITGA2BKDM4EALDH1A1
Hydrochloric Acid SCHEMBL23929053 0.81 PRMT6 (0.57) AGXTITGB3ITGA2BKDM4EALDH1A1
SCHEMBL17115681 0.81 AGXT (0.54) AGXTITGB3ITGA2BKDM4EALDH1A1
SCHEMBL30616970 0.81 ITGB3 (0.50) ITGB3ITGA2BKDM4EALDH1A1MEN1
SCHEMBL15709650 0.80 PRMT6 (0.56) AGXTITGB3ITGA2BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-A SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2019-04-02 CN claimed
CN-109563043-B Substituted pyridines as inhibitors of DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2022-05-31 CN disclosed
CN-104936954-A compounds and methods of use thereof AGIOS PHARMACEUTICALS INC 2015-09-23 CN disclosed