SCHEMBL28030692

SCHEMBL28030692

Cc1nncn1-c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.56
CYP2E1 P05181 2/20 0.56
CYP3A4 P08684 2/20 0.56
ALDH1A1 P00352 3/20 0.43
ALOX12 P18054 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PI4KA P42356 1/20 0.40
PI4K2B Q8TCG2 1/20 0.40
PI4K2A Q9BTU6 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
HTT P42858 1/20 0.40
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA5 P30532 1/20 0.39
CHRNA4 P43681 1/20 0.39
ELANE P08246 1/20 0.39
AR P10275 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10166461 0.80 OPRD1 (0.42) ALDH1A1HTTL3MBTL1MEN1KMT2A
SCHEMBL28100845 0.78 CYP2A6 (0.46) CYP2A6CYP2E1CYP3A4ALDH1A1NPC1
SCHEMBL23576586 0.78 PI4KA (0.46) CYP2A6CYP2E1CYP3A4ALDH1A1NPC1
SCHEMBL6251508 0.77 ALDH1A1 (0.54) CYP2A6CYP2E1CYP3A4ALDH1A1NPC1
SCHEMBL30230906 0.75 CYP2A6 (0.56) CYP2A6CYP2E1CYP3A4ALDH1A1ALOX12
SCHEMBL6251506 0.74 ALDH1A1 (0.51) CYP2A6CYP2E1CYP3A4ALDH1A1NPC1
SCHEMBL3607993 0.73 CYP2A6 (0.55) CYP2A6CYP2E1CYP3A4ALDH1A1ALOX12
SCHEMBL3609259 0.72 CYP2A6 (1.00) CYP2A6CYP2E1CYP3A4ALDH1A1ALOX12
SCHEMBL6756652 0.71 MAPT (0.49) CYP3A4ALDH1A1MEN1KMT2A
SCHEMBL30233195 0.71 MAPK9 (0.40) CYP2A6CYP2E1CYP3A4ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903325-A COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA 2015-09-09 CN disclosed