SCHEMBL28030748

SCHEMBL28030748

CN1CCN(c2ccncc2-n2cc(C(N)=O)cn2)CC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CHEK1 O14757 1/20 0.46
CYP46A1 Q9Y6A2 9/20 0.45
CYP3A4 P08684 1/20 0.44
MELK Q14680 2/20 0.41
BCL2A1 Q16548 1/20 0.40
ATR Q13535 2/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31005773 0.76 CYP3A4 (0.52) KDM4EALDH1A1HSD17B10CHEK1CYP3A4
SCHEMBL17061682 0.76 CYP3A4 (0.49) KDM4EALDH1A1HSD17B10CHEK1CYP3A4
SCHEMBL18228362 0.69 CYP3A4 (0.54) CYP3A4BCL2A1ATR
SCHEMBL15770645 0.68 MAPT (0.63) KDM4EALDH1A1HSD17B10CYP3A4BCL2A1
SCHEMBL16039371 0.68 ADRA2C (0.58) KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL17180151 0.68 CYP46A1 (0.74) KDM4EALDH1A1CYP46A1ATR
SCHEMBL17222774 0.68 CYP46A1 (0.63) CYP46A1
SCHEMBL28332919 0.67 CYP3A4 (0.51) CYP3A4MELKBCL2A1
SCHEMBL31448328 0.67 CHEK1 (0.60) CHEK1MELKATR
SCHEMBL23846557 0.66 F7 (0.54) MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104903325-A COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA 2015-09-09 CN disclosed