Bromide

Bromide

SCHEMBL28030872

Br.Cc1ccc(F)cc1F

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 3/20 0.43
ALDH1A1 P00352 1/20 0.46
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
NFE2L2 Q16236 3/20 0.41
CA3 P07451 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
ATM Q13315 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29367748 0.97
SCHEMBL60954 0.97
Formaldehyde SCHEMBL27818208 0.90 HDAC1 (0.44) ALDH1A1ACHEHDAC1HDAC6PTGS1
SCHEMBL8819778 0.84 KMT2A (0.41) ALDH1A1HDAC1HDAC6PTGS1PTGS2
SCHEMBL29089364 0.80 ACHE (0.48) ALDH1A1ACHEHDAC1HDAC6PTGS1
SCHEMBL26974251 0.80 AKR1C3 (0.54) ALDH1A1MEN1KMT2ANISCH
SCHEMBL29475251 0.79
Bromide SCHEMBL28030910 0.78 CA3 (0.46) ALDH1A1ACHEPTGS1PTGS2CES2
SCHEMBL13906282 0.77 TNKS2 (0.50) ALDH1A1ACHEHDAC1HDAC6NISCH
SCHEMBL12500 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104870422-A Novel amine derivative or salt thereof TOYAMA CHEMICAL CO LTD 2015-08-26 CN disclosed