SCHEMBL28031055

SCHEMBL28031055

Cc1cc(C(N)=O)c(C(F)(F)F)c(C)c1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
POLB P06746 3/20 0.35
LMNA P02545 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.33
CYP3A4 P08684 2/20 0.33
MAPT P10636 3/20 0.33
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
MITF O75030 1/20 0.33
HTT P42858 1/20 0.33
CCR6 P51684 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
BLM P54132 1/20 0.33
PMP22 Q01453 1/20 0.33
PLK1 P53350 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27621172 0.85 POLB (0.38) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL28190932 0.78 ALDH1A1 (0.49) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL28114959 0.77 KMT2A (0.44) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL27621308 0.75 TDP1 (0.39) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL6205026 0.74 TDP1 (0.44) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL4332774 0.74 ALDH1A1 (0.40) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL28114928 0.74 ALDH1A1 (0.37) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL7763285 0.73 ALDH1A1 (0.40) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL21633000 0.72 PARP1 (0.40) ALDH1A1POLBLMNATDP1KMT2A
SCHEMBL28536993 0.72 KMT2A (0.39) ALDH1A1POLBLMNATDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107250110-B Novel compounds as inhibitors of transfection Rearrangement (RET) 葛兰素史克知识产权发展有限公司 2020-04-24 CN disclosed
CN-107250110-A The noval chemical compound of (RET) inhibitor is reset as transfection 葛兰素史克知识产权发展有限公司 2017-10-13 CN disclosed
CN-105051027-A Pyridine derivatives as rearranged during transfection (RET) kinase inhibitors GLAXOSMITHKLINE IP DEV LTD 2015-11-11 CN disclosed