SCHEMBL28031602

SCHEMBL28031602

O=c1cc(-c2ccccc2)oc2cc(OCCBr)cc(O)c12

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.74
ABCB1 P08183 4/20 0.74
MAPT P10636 3/20 0.74
RET P07949 1/20 0.74
KDR P35968 1/20 0.74
CYP1A1 P04798 2/20 0.69
CYP1A2 P05177 2/20 0.69
NPSR1 Q6W5P4 1/20 0.68
CYP3A4 P08684 2/20 0.67
CYP2C9 P11712 2/20 0.67
CYP2C19 P33261 2/20 0.67
ABCG2 Q9UNQ0 2/20 0.67
NPC1 O15118 1/20 0.67
TSHR P16473 1/20 0.67
KDM4E B2RXH2 1/20 0.66
MEN1 O00255 1/20 0.66
GABRP O00591 1/20 0.66
GABRD O14764 1/20 0.66
CA12 O43570 1/20 0.66
AKR1B10 O60218 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12792587 0.94 EGFR (0.72) EGFRABCB1MAPTRETKDR
SCHEMBL13186952 0.92 EGFR (0.69) EGFRABCB1MAPTRETKDR
SCHEMBL10025658 0.90 MAPT (0.77) EGFRABCB1MAPTRETKDR
SCHEMBL12678185 0.87 EGFR (0.80) EGFRABCB1MAPTRETKDR
SCHEMBL974548 0.85 MAPT (1.00) EGFRABCB1MAPTRETKDR
SCHEMBL30376285 0.85 MAPT (1.00) EGFRABCB1MAPTRETKDR
SCHEMBL433900 0.84 EGFR (0.71) EGFRABCB1MAPTRETKDR
SCHEMBL24882669 0.83 EGFR (0.78) EGFRABCB1MAPTRETKDR
SCHEMBL16823312 0.83 EGFR (0.70) EGFRABCB1MAPTRETKDR
SCHEMBL431393 0.82 EGFR (0.69) EGFRRETKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103242309-B A kind of chrysin thiazole derivative and its preparation method and application NANJING UNIVERSITY (CN) 2015-08-05 CN disclosed